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LIT-PCBA

Literature-curated dose-response PubChem BioAssay set; 15 targets with unbiased actives/inactives.
Composite score: 80.8

Rubric (1–5 per criterion)

rigor
5/5
coverage
3/5
maintenance
2/5
adoption
4/5
quality
5/5
accessibility
5/5
industry_relevance
4/5

Metadata

Stages
Hit ID
Modalities
small-molecule
Task types
virtual-screening
License
CC-BY
First release
2020-03
Last updated
2023-06
Flags
none

Size & scope

Primary paper

Title
LIT-PCBA: An Unbiased Data Set for Machine Learning and Virtual Screening
Authors
Tran-Nguyen VK, Jacquemard C, Rognan D
Year
2020
DOI / arXiv
10.1021/acs.jcim.0c00155
Citations
310

Links

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Experts (primary authors / maintainers)

Groups (host labs / companies / consortia)

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Notes (honest caveats)

Much fairer than DUD-E; small target count limits coverage.